Skip To Main Content
Lilly
Menu closed
Lilly
  • Account Login / Register
  • Medical Home
    • Medical Information
  • Medical Education
  • Science
Ask Lilly

We're here to help.

Chat
Chat with us
Question Contact Us
Expand contact lilly
Lilly

You are now leaving the Lilly Medical website

The link you clicked on will take you to a site maintained by a third party, which is solely responsible for its content. Lilly USA, LLC does not control, influence, or endorse this site, and the opinions, claims, or comments expressed on this site should not be attributed to Lilly USA, LLC. Lilly USA, LLC is not responsible for the privacy policy of any third-party websites. We encourage you to read the privacy policy of every website you visit.
Click "Continue" to proceed or "Return" to return to Lilly Medical

  1. Medical Information Right
  2. Obesity Right
  3. Foundayo (orforglipron) tablet Right
  4. What is the approved dosing for Foundayo™ (orforglipron) for weight management?
Search Foundayo (type in keywords)
Search Medical Information

If you wish to report an adverse event or product complaint, please call 1-800-LILLYRX (1-800-545-5979)

Loading icon

Foundayo ™ (orforglipron) tablet

0.8 mg / 2.5 mg / 5.5 mg / 9 mg / 14.5 mg / 17.2 mg

Full Prescribing Information

This information is provided in response to your request. Resources may contain information about doses, uses, formulations and populations different from product labeling. See Prescribing Information above, if applicable.

What is the approved dosing for Foundayo™ (orforglipron) for weight management?

The starting dose is 0.8 mg once daily. After ≥30 days, increase to 2.5 mg once daily. After ≥30 days, increase to 5.5 mg once daily. After ≥30 days, the dosage may be increased to 9.0, 14.5, or 17.2 mg once daily. The maximum dose is 17.2 mg once daily.

US_cFAQ_OFG600B_APPROVED_DOSING_WM
US_cFAQ_OFG600B_APPROVED_DOSING_WMen-US

See important safety information, including boxed warning, in the attached prescribing information.

Content Overview 

What Is the Approved Dosing and Method of Administration of Orforglipron for Weight Management?

  • Orforglipron Recommended Dosage Escalation 

Are There Any Recommended Dose Modifications for Orforglipron?

  • Dosing Considerations in Patients With Hepatic Impairment 
  • Orforglipron Dosage Considerations With Concomitant CYP3A4 Inhibitors and CYP3A4 Inducers
    • Dosage Considerations With Strong CYP3A4 Inhibitors 
    • Dosage Considerations With Strong or Moderate CYP3A4 Inducers
  • Additional Considerations 

Enclosed Prescribing Information

Reference

What Is the Approved Dosing and Method of Administration of Orforglipron for Weight Management?

Orforglipron is indicated in combination with a reduced-calorie diet and increased physical activity to reduce excess body weight and maintain weight reduction long term in adults with

  • obesity, or
  • overweight in the presence of at least one weight-related comorbid condition.1

In the United States, orforglipron is available in tablet form in dosages of

  • 0.8 mg
  • 2.5 mg
  • 5.5 mg
  • 9 mg
  • 14.5 mg, and 
  • 17.2 mg.1

Take orforglipron orally once daily, with or without food.1

Swallow tablets whole. Do not break, crush, or chew.1

Do not take more than one tablet per day.1

Orforglipron Recommended Dosage Escalation 

Follow the orforglipron starting dose and escalation described below to reduce the risk of gastrointestinal adverse reactions.1

  • The starting dosage is 0.8 mg orally once daily. After at least 30 days on the 0.8 mg, increase the dosage to 2.5 mg once daily.1
  • After at least 30 days on the 2.5 mg dosage, increase the dosage to 5.5 mg once daily.1
  • The dosage may be increased to the next dosage level (9 mg, 14.5 mg, or 17.2 mg once daily) after at least 30 days on the current dosage, based on treatment response and tolerability.1
  • The maximum dosage of orforglipron is 17.2 mg once daily.1

Are There Any Recommended Dose Modifications for Orforglipron?

The following intrinsic factors do not have a clinically relevant effect on the pharmacokinetics of orforglipron including

  • age (18 to 92 years old)
  • sex
  • race (White, Asian, Black or African American, American Indian, Multiracial, or Hawaiian Pacific Islander)
  • ethnicity (Hispanic, Non-Hispanic)
  • body weight (56.4 to 227 kg), and
  • renal impairment (estimated glomerular filtration rate 27.8 to 156 L/min/1.73 m2).1

The orforglipron prescribing information does not include dosing modification recommendations based on these factors.1

Dosing Considerations in Patients With Hepatic Impairment 

Orforglipron is not recommended for use in patients with severe hepatic impairment (Child-Pugh Class C).1

No dosage adjustment of orforglipron is recommended in patients with mild or moderate hepatic impairment (Child-Pugh Class A and B, respectively).1

Orforglipron Dosage Considerations With Concomitant CYP3A4 Inhibitors and CYP3A4 Inducers

Orforglipron dose adjustment may be required to manage interactions with some concomitant medications.1

Dosage Considerations With Strong CYP3A4 Inhibitors 

Avoid concomitant use of orforglipron with strong cytochrome P450 3A4 (CYP3A4) inhibitors that also inhibit organic anion transporting polypeptide 1B (OATP1B) (eg, ritonavir).1

The maximum dosage is orforglipron 9 mg once daily when used concomitantly with a strong CYP3A4 inhibitor.1

Dosage Considerations With Strong or Moderate CYP3A4 Inducers

Avoid concomitant use of orforglipron with strong CYP3A4 inducers.1

Monitor orforglipron effectiveness and escalate dosage as needed when used concomitantly with moderate CYP3A4 inducers.1

Additional Considerations 

Eli Lilly and Company cannot provide dosing recommendations that go beyond those in the approved label, as these treatment scenarios have likely not been studied.

There is no information available on dosage strengths beyond the approved doses or on dosing intervals longer than once daily, as these have not been evaluated in clinical studies.

Enclosed Prescribing Information

FOUNDAYO™ (orforglipron) tablets, for oral use, Lilly

Reference

1Foundayo [package insert]. Indianapolis, IN: Eli Lilly and Company; 2026.

Date of Last Review: April 01, 2026

Are you satisfied with this content?

Can't find what you're looking for? Contact us for answers to your medical questions.

  • Copyright
  • Terms of Use
  • Privacy Statement
  • Consumer Health Privacy Notice
  • Accessibility Statement
  • Sitemap

    This site is intended for US Healthcare Professionals only.

    4.0.53 05/2026 | GLOOTH00001 04/2015 | © Lilly USA, LLC 2026. All rights reserved.

    Product names listed above are trademarks or registered trademarks owned by or licensed to Eli Lilly and Company, its subsidiaries, or affiliates

    California Consumer Privacy Act (CCPA) Opt-Out Icon Your Privacy Choices
    Cookie Settings
    facebook twitter linkedin
    visit www.phactmi.org
    Lilly